AMPHOTERICIN B, IV

  • Amphotericin B, IV, 0.7–­1 mg/kg daily, dose and duration of therapy depend on indication for use and infecting organism.
    • Reconstitue in 5% dextrose water only (as incompatibile with saline solution).
    • Administer over a period of 2–6 hours.
    • Ensure adequate hydration to minimise the risk of nephrotoxicity.

Monitoring

  • Serum potassium, magnesium and creatinine (baseline and twice weekly). Monitoring of serum potassium and creatinine should occur more frequently in neutropenic patients (3 times a week).
  • Monitor haemoglobin (baseline and weekly).
  • Careful attention to fluid monitoring of intake and output.
  • For management of hypokalaemia, see section 7.2.2: Hypokalaemia.

Management of elevated creatinine

If creatinine increases by ≥2 fold from baseline value, either omit an amphotericin B dose, or increase pre-hydration to 1 litre 8 hourly.

  • Once improved, restart at 0.7 mg/kg daily and consider alternate day amphotericin B.
  • If creatinine remains elevated i.e. ≥2 fold from baseline value, discontinue amphotericin B and continue with fluconazole, oral, 800 mg daily (for fungal infections known to be responsive to fluconazole, e.g. Cryptococcus).

(Adapted from: WHO. Rapid advice: diagnosis, prevention and management of cryptococcal disease in HIV-infected adults, adolescents and children: Prevention, monitoring and management of amphotericin B toxicity. 2011 [Online] [Accessed March 2016] http://www.ncbi.nlm.nih.gov/books/NBK299520/pdf/Bookshelf_NBK299520.pdf